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药效评价Combined anti CXC receptors 1 and 2 therapy is a promising anti-inflammatory treatment for respiratory diseases by reducing neutrophil migration and activation.

期刊:Pulmonary pharmacology & therapeutics发表年份:2015作者:A Planagumà; T Domènech; M Pont; E Calama; V García-González; R López; M Aulí; M López; S Fonquerna; I Ramos; J de Alba; A Nueda; N Prats; V Segarra; M Miralpeix; M D Lehner

药效评价Pharmacological lineage analysis revealed the binding affinity of broad-spectrum substance P antagonists to receptors for gonadotropin-releasing peptide.

期刊:European journal of pharmacology发表年份:2015作者:Kazune Arai; Aki Kashiwazaki; Yoko Fujiwara; Hiroyoshi Tsuchiya; Nobuya Sakai; Katsushi Shibata; Taka-aki Koshimizu

药效评价Pharmacological characterization of the newly synthesized 5-amino-N-butyl-2-(4-ethoxyphenoxy)-benzamide hydrochloride (BED) as a potent NCX3 inhibitor that worsens anoxic injury in cortical neurons, organotypic hippocampal cultures, and ischemic brai

期刊:ACS chemical neuroscience发表年份:2015作者:Agnese Secondo; Giuseppe Pignataro; Paolo Ambrosino; Anna Pannaccione; Pasquale Molinaro; Francesca Boscia; Maria Cantile; Ornella Cuomo; Alba Esposito; Maria Josè Sisalli; Antonella Scorziello; Natascia Guida; Serenella Anzilotti; Ferdinando Fiorino

药效评价A potent and selective C-11 labeled PET tracer for imaging sphingosine-1-phosphate receptor 2 in the CNS demonstrates sexually dimorphic expression.

期刊:Organic & biomolecular chemistry发表年份:2015作者:Xuyi Yue; Hongjun Jin; Hui Liu; Adam J Rosenberg; Robyn S Klein; Zhude Tu