郑州微飒生物科技有限责任公司 咨询热线:0371-88821766
行业动态

行业动态

追踪行业前沿,洞察产业趋势

药效评价Discovery, synthesis, and molecular pharmacology of selective positive allosteric modulators of the δ-opioid receptor.

期刊:Journal of medicinal chemistry发表年份:2015作者:Neil T Burford; Kathryn E Livingston; Meritxell Canals; Molly R Ryan; Lauren M L Budenholzer; Ying Han; Yi Shang; John J Herbst; Jonathan O'Connell; Martyn Banks; Litao Zhang; Marta Filizola; Daniel L Bassoni; Tom S Wehrman; Arthur Christopoulos; Joh

药效评价A solid-phase combinatorial approach for indoloquinolizidine-peptides with high affinity at D(1) and D(2) dopamine receptors.

期刊:European journal of medicinal chemistry发表年份:2015作者:Anabel Molero; Marc Vendrell; Jordi Bonaventura; Julian Zachmann; Laura López; Leonardo Pardo; Carme Lluis; Antoni Cortés; Fernando Albericio; Vicent Casadó; Miriam Royo

药效评价Quantitative Measurement of GPCR Endocytosis via Pulse-Chase Covalent Labeling.

期刊:PloS one发表年份:2015作者:Hidetoshi Kumagai; Yuichi Ikeda; Yoshihiro Motozawa; Mitsuhiro Fujishiro; Tomohisa Okamura; Keishi Fujio; Hiroaki Okazaki; Seitaro Nomura; Norifumi Takeda; Mutsuo Harada; Haruhiro Toko; Eiki Takimoto; Hiroshi Akazawa; Hiroyuki Morita; Jun-ichi Suzuki

药效评价Co-operative binding assay for the characterization of mGlu4 allosteric modulators.

期刊:Neuropharmacology发表年份:2015作者:Pekka Poutiainen; Kun-Eek Kil; Zhaoda Zhang; Darshini Kuruppu; Bakhos Tannous; Anna-Liisa Brownell