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药效评价Lipoic-based TRPA1/TRPV1 antagonist to treat orofacial pain.

期刊:ACS chemical neuroscience发表年份:2015作者:Roberta Gualdani; Stefania Ceruti; Giulia Magni; Davide Merli; Lorenzo Di Cesare Mannelli; Oscar Francesconi; Barbara Richichi; Giancarlo la Marca; Carla Ghelardini; Maria Rosa Moncelli; Cristina Nativi

药效评价Exposure to Δ9-Tetrahydrocannabinol Impairs the Differentiation of Human Monocyte-derived Dendritic Cells and their Capacity for T cell Activation.

期刊:Journal of neuroimmune pharmacology : the official journal of the Society on NeuroImmune Pharmacology发表年份:2015作者:Michael D Roth; Julie T Castaneda; Sylvia M Kiertscher

药效评价Discovery of (R)-1-(3-((2-chloro-4-(((2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethyl)amino)methyl)-5-methoxyphenyl)amino)-3-oxopropyl)piperidin-4-yl [1,1'-biphenyl]-2-ylcarbamate (TD-5959, GSK961081, batefenterol): first-in-class dual ph

期刊:Journal of medicinal chemistry发表年份:2015作者:Adam D Hughes; Yan Chen; Sharath S Hegde; Jeffrey R Jasper; Sarah Jaw-Tsai; Tae-Weon Lee; Alexander McNamara; M Teresa Pulido-Rios; Tod Steinfeld; Mathai Mammen

药效评价Cell-based and virtual fragment screening for adrenergic α2C receptor agonists.

期刊:Bioorganic & medicinal chemistry发表年份:2015作者:Edit Szőllősi; Amrita Bobok; László Kiss; Márton Vass; Dalma Kurkó; Sándor Kolok; András Visegrády; György M Keserű