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药效评价A Novel Modulator of Kv3 Potassium Channels Regulates the Firing of Parvalbumin-Positive Cortical Interneurons.

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2015作者:Marcelo D Rosato-Siri; Erika Zambello; Chiara Mutinelli; Nicoletta Garbati; Roberto Benedetti; Laura Aldegheri; Francesca Graziani; Caterina Virginio; Giuseppe Alvaro; Charles H Large

药效评价Characterization of V0162, a new long-acting antagonist at human M3 muscarinic acetylcholine receptors.

期刊:Pharmacological research发表年份:2015作者:Peter Heusler; Didier Cussac; Emmanuel Naline; Stéphanie Tardif; Thierry Clerc; Philippe Devillier

药效评价Novel Synthesis and Pharmacological Characterization of NOP Receptor Agonist 8-[(1S,3aS)-2,3,3a,4,5,6-Hexahydro-1H-phenalen-1-yl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one (Ro 64-6198).

期刊:ACS chemical neuroscience发表年份:2015作者:Steven D Chang; Lawrence E Brieaddy; Joseph D Harvey; Anita H Lewin; S Wayne Mascarella; Herbert H Seltzman; P Anantha Reddy; Ann M Decker; Charles J McElhinny; Desong Zhong; Elisha E Peterson; Hernán A Navarro; Michael R Bruchas; F Ivy Carroll

药效评价Optimization of on-resin palladium-catalyzed Sonogashira cross-coupling reaction for peptides and its use in a structure-activity relationship study of a class B GPCR ligand.

期刊:European journal of medicinal chemistry发表年份:2015作者:Ngoc-Duc Doan; Mathilde Poujol de Molliens; Myriam Létourneau; Alain Fournier; David Chatenet