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药效评价Differential impact of amino acid substitutions on critical residues of the human glucagon-like peptide-1 receptor involved in peptide activity and small-molecule allostery.

期刊：The Journal of pharmacology and experimental therapeutics发表年份：2015作者：Cassandra Koole; Denise Wootten; John Simms; Laurence J Miller; Arthur Christopoulos; Patrick M Sexton
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药效评价Discovery of the first small-molecule opioid pan antagonist with nanomolar affinity at mu, delta, kappa, and nociceptin opioid receptors.

期刊：ACS chemical neuroscience发表年份：2015作者：Nurulain T Zaveri; V Blair Journigan; Willma E Polgar
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药效评价Design, syntheses, structure-activity relationships and docking studies of coumarin derivatives as novel selective ligands for the CB2 receptor.

期刊：European journal of medicinal chemistry发表年份：2015作者：Shuang Han; Fei-Fei Zhang; Hai-Yan Qian; Li-Li Chen; Jian-Bin Pu; Xin Xie; Jian-Zhong Chen
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药效评价Detection of new biased agonists for the serotonin 5-HT2A receptor: modeling and experimental validation.

期刊：Molecular pharmacology发表年份：2015作者：Maria Martí-Solano; Alba Iglesias; Gianni de Fabritiis; Ferran Sanz; José Brea; M Isabel Loza; Manuel Pastor; Jana Selent
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