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药效评价BU08073 a buprenorphine analogue with partial agonist activity at μ-receptors in vitro but long-lasting opioid antagonist activity in vivo in mice.

期刊:British journal of pharmacology发表年份:2015作者:T V Khroyan; J Wu; W E Polgar; G Cami-Kobeci; N Fotaki; S M Husbands; L Toll

药效评价Is the acetylcholine-regulated inwardly rectifying potassium current a viable antiarrhythmic target? Translational discrepancies of AZD2927 and A7071 in dogs and humans.

期刊:Europace : European pacing, arrhythmias, and cardiac electrophysiology : journal of the working groups on cardiac pacing, arrhythmias, and cardiac cellular electrophysiology of the European Society of Cardiology发表年份:2015作者:Håkan Walfridsson; Ole-Gunnar Anfinsen; Anders Berggren; Lars Frison; Steen Jensen; Gunilla Linhardt; Ann-Christin Nordkam; Monika Sundqvist; Leif Carlsson

药效评价Pharmacological and signalling properties of a D2-like dopamine receptor (Dop3) in Tribolium castaneum.

期刊:Insect biochemistry and molecular biology发表年份:2015作者:Heleen Verlinden; Rut Vleugels; Rik Verdonck; Elodie Urlacher; Jozef Vanden Broeck; Alison Mercer

药效评价Rational design of partial agonists for the muscarinic m1 acetylcholine receptor.

期刊:Journal of medicinal chemistry发表年份:2015作者:Xinyu Chen; Jessika Klöckner; Janine Holze; Cornelia Zimmermann; Wiebke K Seemann; Ramona Schrage; Andreas Bock; Klaus Mohr; Christian Tränkle; Ulrike Holzgrabe; Michael Decker