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药效评价Molecular hybridization yields triazole bronchodilators for the treatment of COPD.

期刊:Bioorganic & medicinal chemistry letters发表年份:2015作者:Lyn H Jones; Jane Burrows; Neil Feeder; Paul Glossop; Kim James; Rhys M Jones; Amy S Kenyon; Sheena Patel; Dannielle F Roberts; Matthew D Selby; Ross S Strang; Emilio F Stuart; Michael A Trevethick; Jessica Watson; Karen N Wright; Nick Clarke

药效评价Fragment-Based Discovery of Subtype-Selective Adenosine Receptor Ligands from Homology Models.

期刊:Journal of medicinal chemistry发表年份:2015作者:Anirudh Ranganathan; Leigh A Stoddart; Stephen J Hill; Jens Carlsson

药效评价mGlu2 Receptor Agonism, but Not Positive Allosteric Modulation, Elicits Rapid Tolerance towards Their Primary Efficacy on Sleep Measures in Rats.

期刊:PloS one发表年份:2015作者:Abdallah Ahnaou; Hilde Lavreysen; Gary Tresadern; Jose M Cid; Wilhelmus H Drinkenburg

药效评价The molecular mechanism of photochemical internalization of cell penetrating peptide-cargo-photosensitizer conjugates.

期刊:Scientific reports发表年份:2015作者:Takashi Ohtsuki; Shunya Miki; Shouhei Kobayashi; Tokuko Haraguchi; Eiji Nakata; Kazutaka Hirakawa; Kensuke Sumita; Kazunori Watanabe; Shigetoshi Okazaki