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药效评价Biased Agonism of Endogenous Opioid Peptides at the μ-Opioid Receptor.

期刊：Molecular pharmacology发表年份：2015作者：Georgina L Thompson; J Robert Lane; Thomas Coudrat; Patrick M Sexton; Arthur Christopoulos; Meritxell Canals
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药效评价Primary Macrophage Chemotaxis Induced by Cannabinoid Receptor 2 Agonists Occurs Independently of the CB2 Receptor.

期刊：Scientific reports发表年份：2015作者：Lewis Taylor; Ivy Christou; Theodore S Kapellos; Alice Buchan; Maximillian H Brodermann; Matteo Gianella-Borradori; Angela Russell; Asif J Iqbal; David R Greaves
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药效评价Structure-activity study of N-((trans)-4-(2-(7-cyano-3,4-dihydroisoquinolin-2(1H)-yl)ethyl)cyclohexyl)-1H-indole-2-carboxamide (SB269652), a bitopic ligand that acts as a negative allosteric modulator of the dopamine D2 receptor.

期刊：Journal of medicinal chemistry发表年份：2015作者：Jeremy Shonberg; Christopher Draper-Joyce; Shailesh N Mistry; Arthur Christopoulos; Peter J Scammells; J Robert Lane; Ben Capuano
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药效评价Identification of the First Highly Subtype-Selective Inhibitor of Human GABA Transporter GAT3.

期刊：ACS chemical neuroscience发表年份：2015作者：Maria Damgaard; Anas Al-Khawaja; Stine B Vogensen; Andreas Jurik; Maarten Sijm; Maria E K Lie; Mathias I Bæk; Emil Rosenthal; Anders A Jensen; Gerhard F Ecker; Bente Frølund; Petrine Wellendorph; Rasmus P Clausen
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