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药效评价Pharmacology of basimglurant (RO4917523, RG7090), a unique metabotropic glutamate receptor 5 negative allosteric modulator in clinical development for depression.

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2015作者:Lothar Lindemann; Richard H Porter; Sebastian H Scharf; Basil Kuennecke; Andreas Bruns; Markus von Kienlin; Anthony C Harrison; Axel Paehler; Christoph Funk; Andreas Gloge; Manfred Schneider; Neil J Parrott; Liudmila Polonchuk; Urs Niederhauser; Step

药效评价Introduction of germline residues improves the stability of anti-HIV mAb 2G12-IgM.

期刊:Biochimica et biophysica acta发表年份:2015作者:Veronika Chromikova; Alexander Mader; Stefan Hofbauer; Christoph Göbl; Tobias Madl; Johannes S Gach; Stefan Bauernfried; Paul G Furtmüller; Donald N Forthal; Lukas Mach; Christian Obinger; Renate Kunert

药效评价Novel halogenated derivates of JWH-018: Behavioral and binding studies in mice.

期刊:Neuropharmacology发表年份:2015作者:A Vigolo; A Ossato; C Trapella; F Vincenzi; C Rimondo; C Seri; K Varani; G Serpelloni; M Marti

药效评价Discovery of a potent, orally available dual CysLT₁ and CysLT₂ antagonist with dicarboxylic acid.

期刊:Bioorganic & medicinal chemistry发表年份:2015作者:Satoshi Itadani; Shinya Takahashi; Masaki Ima; Tetsuya Sekiguchi; Yoshiyuki Aratani; Hiromu Egashira; Naoya Matsumura; Atsuto Inoue; Yasuo Yonetomi; Manabu Fujita; Yoshisuke Nakayama; Jun Takeuchi