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药效评价Discovery and mapping of an intracellular antagonist binding site at the chemokine receptor CCR2.

期刊:Molecular pharmacology发表年份:2014作者:Annelien J M Zweemer; Julia Bunnik; Margo Veenhuizen; Fabiana Miraglia; Eelke B Lenselink; Maris Vilums; Henk de Vries; Arthur Gibert; Stefanie Thiele; Mette M Rosenkilde; Adriaan P IJzerman; Laura H Heitman

药效评价Mechanistic insights into allosteric structure-function relationships at the M1 muscarinic acetylcholine receptor.

期刊:The Journal of biological chemistry发表年份:2014作者:Alaa Abdul-Ridha; J Robert Lane; Shailesh N Mistry; Laura López; Patrick M Sexton; Peter J Scammells; Arthur Christopoulos; Meritxell Canals

药效评价Complex relationships between substrate sequence and sensitivity to alterations in γ-secretase processivity induced by γ-secretase modulators.

期刊:Biochemistry发表年份:2014作者:Joo In Jung; Yong Ran; Pedro E Cruz; Awilda M Rosario; Thomas B Ladd; Thomas L Kukar; Edward H Koo; Kevin M Felsenstein; Todd E Golde

药效评价Inhibition of HERG potassium channels by domiphen bromide and didecyl dimethylammonium bromide.

期刊:European journal of pharmacology发表年份:2014作者:Yan Long; Wanjuan Chen; Zuoxian Lin; Hongmao Sun; Menghang Xia; Wei Zheng; Zhiyuan Li