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药效评价Blocking metabotropic glutamate receptor subtype 7 (mGlu7) via the Venus flytrap domain (VFTD) inhibits amygdala plasticity, stress, and anxiety-related behavior.

期刊:The Journal of biological chemistry发表年份:2014作者:Christine E Gee; Daniel Peterlik; Christoph Neuhäuser; Rochdi Bouhelal; Klemens Kaupmann; Grit Laue; Nicole Uschold-Schmidt; Dominik Feuerbach; Kaspar Zimmermann; Silvio Ofner; John F Cryan; Herman van der Putten; Markus Fendt; Ivo Vranesic; Ralf Gla

药效评价Na+/H+ exchanger 1 is regulated via its lipid-interacting domain, which functions as a molecular switch: a pharmacological approach using indolocarbazole compounds.

期刊:Molecular pharmacology发表年份:2014作者:Naoko Shimada-Shimizu; Takashi Hisamitsu; Tomoe Y Nakamura; Noriaki Hirayama; Shigeo Wakabayashi

药效评价Mefloquine and psychotomimetics share neurotransmitter receptor and transporter interactions in vitro.

期刊:Psychopharmacology发表年份:2014作者:Aaron Janowsky; Amy J Eshleman; Robert A Johnson; Katherine M Wolfrum; David J Hinrichs; Jongtae Yang; T Mark Zabriskie; Martin J Smilkstein; Michael K Riscoe

药效评价Brexpiprazole I: in vitro and in vivo characterization of a novel serotonin-dopamine activity modulator.

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2014作者:Kenji Maeda; Haruhiko Sugino; Hitomi Akazawa; Naoki Amada; Jun Shimada; Takashi Futamura; Hiroshi Yamashita; Nobuaki Ito; Robert D McQuade; Arne Mørk; Alan L Pehrson; Morten Hentzer; Vibeke Nielsen; Christoffer Bundgaard; Jørn Arnt; Tine Bryan Stensb