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药效评价Different efficacy of adenosine and NECA derivatives at the human A3 adenosine receptor: insight into the receptor activation switch.

期刊:Biochemical pharmacology发表年份:2014作者:Diego Dal Ben; Michela Buccioni; Catia Lambertucci; Sonja Kachler; Nico Falgner; Gabriella Marucci; Ajiroghene Thomas; Gloria Cristalli; Rosaria Volpini; Karl-Norbert Klotz

药效评价Pharmacologic characterization of GSK-961081 (TD-5959), a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2014作者:Sharath S Hegde; Adam D Hughes; Yan Chen; Tod Steinfeld; Jeffrey R Jasper; Tae-Weon Lee; Alexander McNamara; William J Martin; M Teresa Pulido-Rios; Mathai Mammen

药效评价Neurophysiologic and antipsychotic profiles of TASP0433864, a novel positive allosteric modulator of metabotropic glutamate 2 receptor.

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2014作者:Tetsuaki Hiyoshi; Toshiyuki Marumo; Hirohiko Hikichi; Yasumitsu Tomishima; Hiroki Urabe; Tomoko Tamita; Izumi Iida; Akito Yasuhara; Jun-ichi Karasawa; Shigeyuki Chaki

药效评价TRR469, a potent A(1) adenosine receptor allosteric modulator, exhibits anti-nociceptive properties in acute and neuropathic pain models in mice.

期刊:Neuropharmacology发表年份:2014作者:Fabrizio Vincenzi; Martina Targa; Romeo Romagnoli; Stefania Merighi; Stefania Gessi; Pier Giovanni Baraldi; Pier Andrea Borea; Katia Varani