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药效评价Radiosynthesis and evaluation of an 18F-labeled positron emission tomography (PET) radioligand for metabotropic glutamate receptor subtype 4 (mGlu4).

期刊:Journal of medicinal chemistry发表年份:2014作者:Kun-Eek Kil; Pekka Poutiainen; Zhaoda Zhang; Aijun Zhu; Ji-Kyung Choi; Kimmo Jokivarsi; Anna-Liisa Brownell

药效评价Synthesis and κ-opioid receptor activity of furan-substituted salvinorin A analogues.

期刊:Journal of medicinal chemistry发表年份:2014作者:Andrew P Riley; Chad E Groer; David Young; Amy W Ewald; Bronwyn M Kivell; Thomas E Prisinzano

药效评价The phosphoinositide-dependent protein kinase 1 inhibitor, UCN-01, induces fragmentation: possible role of metalloproteinases.

期刊:European journal of pharmacology发表年份:2014作者:Rocío Alcántara-Hernández; Aurelio Hernández-Méndez; J Adolfo García-Sáinz

药效评价Orally active opioid μ/δ dual agonist MGM-16, a derivative of the indole alkaloid mitragynine, exhibits potent antiallodynic effect on neuropathic pain in mice.

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2014作者:Kenjiro Matsumoto; Minoru Narita; Naotaka Muramatsu; Terumi Nakayama; Kaori Misawa; Mariko Kitajima; Kimihito Tashima; Lakshmi A Devi; Tsutomu Suzuki; Hiromitsu Takayama; Syunji Horie