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药效评价Potential of 2-hydroxy-3-phenylsulfanylmethyl-[1,4]-naphthoquinones against Leishmania (L.) infantum: biological activity and structure-activity relationships.

期刊:PloS one发表年份:2014作者:Erika G Pinto; Isabela O Santos; Thomas J Schmidt; Samanta E T Borborema; Vitor F Ferreira; David R Rocha; Andre G Tempone

药效评价Effects of the neuropeptide S receptor antagonist RTI-118 on abuse-related facilitation of intracranial self-stimulation produced by cocaine and methylenedioxypyrovalerone (MDPV) in rats.

期刊:European journal of pharmacology发表年份:2014作者:Julie S Bonano; Scott P Runyon; Carla Hassler; Richard A Glennon; S Stevens Negus

药效评价Synthesis and biological evaluation of a novel series of heterobivalent muscarinic ligands based on xanomeline and 1-[3-(4-butylpiperidin-1-yl)propyl]-1,2,3,4-tetrahydroquinolin-2-one (77-LH-28-1).

期刊:Journal of medicinal chemistry发表年份:2014作者:Alessandro Bonifazi; Hideaki Yano; Fabio Del Bello; Aniket Farande; Wilma Quaglia; Riccardo Petrelli; Rosanna Matucci; Marta Nesi; Giulio Vistoli; Sergi Ferré; Alessandro Piergentili

药效评价Preclinical pharmacology, ocular tolerability and ocular hypotensive efficacy of a novel non-peptide bradykinin mimetic small molecule.

期刊:Experimental eye research发表年份:2014作者:Najam A Sharif; Linya Li; Parvaneh Katoli; Shouxi Xu; James Veltman; Byron Li; Daniel Scott; Martin Wax; Juana Gallar; Carmen Acosta; Carlos Belmonte