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药效评价Discovery and characterization of a G protein-biased agonist that inhibits β-arrestin recruitment to the D2 dopamine receptor.

期刊:Molecular pharmacology发表年份:2014作者:R Benjamin Free; Lani S Chun; Amy E Moritz; Brittney N Miller; Trevor B Doyle; Jennie L Conroy; Adrian Padron; Julie A Meade; Jingbo Xiao; Xin Hu; Andrés E Dulcey; Yang Han; Lihua Duan; Steve Titus; Melanie Bryant-Genevier; Elena Barnaeva; Marc Ferre

药效评价Functionally selective dopamine D₂, D₃ receptor partial agonists.

期刊:Journal of medicinal chemistry发表年份:2014作者:Dorothee Möller; Ralf C Kling; Marika Skultety; Kristina Leuner; Harald Hübner; Peter Gmeiner

药效评价Verification of a new biocompatible single-use film formulation with optimized additive content for multiple bioprocess applications.

期刊:Biotechnology progress发表年份:2014作者:Elke Jurkiewicz; Ute Husemann; Gerhard Greller; Magali Barbaroux; Christel Fenge

药效评价An allosteric switch for pro-HGF/Met signaling using zymogen activator peptides.

期刊:Nature chemical biology发表年份:2014作者:Kyle E Landgraf; Micah Steffek; Clifford Quan; Jeffrey Tom; Christine Yu; Lydia Santell; Henry R Maun; Charles Eigenbrot; Robert A Lazarus