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药效评价Cyclosporine A and PSC833 inhibit ABCA1 function via direct binding.

期刊:Biochimica et biophysica acta发表年份:2013作者:Kohjiro Nagao; Minami Maeda; Noralyn B Mañucat; Kazumitsu Ueda

药效评价Discovery of novel α₁-adrenoceptor ligands based on the antipsychotic sertindole suitable for labeling as PET ligands.

期刊:Bioorganic & medicinal chemistry发表年份:2013作者:Morten Jørgensen; Pernille N Jørgensen; Claus T Christoffersen; Klaus G Jensen; Thomas Balle; Benny Bang-Andersen

药效评价Polar solvents decrease the viscosity of high concentration IgG1 solutions through hydrophobic solvation and interaction: formulation and biocompatibility considerations.

期刊:Journal of pharmaceutical sciences发表年份:2013作者:Tim J Kamerzell; Amanda L Pace; Megan Li; Dimitry M Danilenko; Michelle McDowell; Yatin R Gokarn; Y John Wang

药效评价Modulation of cytochromes P450 with xanthone-based molecules: from aromatase to aldosterone synthase and steroid 11β-hydroxylase inhibition.

期刊:Journal of medicinal chemistry发表年份:2013作者:Silvia Gobbi; Qingzhong Hu; Matthias Negri; Christina Zimmer; Federica Belluti; Angela Rampa; Rolf W Hartmann; Alessandra Bisi