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药效评价Asymmetric total synthesis and identification of tetrahydroprotoberberine derivatives as new antipsychotic agents possessing a dopamine D(1), D(2) and serotonin 5-HT(1A) multi-action profile.

期刊:Bioorganic & medicinal chemistry发表年份:2013作者:Haifeng Sun; Liyuan Zhu; Huicui Yang; Wangke Qian; Lin Guo; Shengbin Zhou; Bo Gao; Zeng Li; Yu Zhou; Hualiang Jiang; Kaixian Chen; Xuechu Zhen; Hong Liu

药效评价Protein expression, biochemical pharmacology of signal transduction, and relation to intraocular pressure modulation by bradykinin B₂ receptors in ciliary muscle.

期刊:Molecular vision发表年份:2013作者:Najam A Sharif; Shouxi Xu; Linya Li; Parvaneh Katoli; Curtis R Kelly; Yu Wang; Shutong Cao; Rajkumar Patil; Shahid Husain; Laura Klekar; Daniel Scott

药效评价In pursuit of synthetic modulators for the orphan retina-specific nuclear receptor NR2E3.

期刊:Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics发表年份:2013作者:Qiong Qin; Anna Knapinska; Nicoleta Dobri; Franck Madoux; Peter Chase; Peter Hodder; Konstantin Petrukhin

药效评价In vitro pharmacological characterization of vilanterol, a novel long-acting β2-adrenoceptor agonist with 24-hour duration of action.

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2013作者:Robert J Slack; Victoria J Barrett; Valerie S Morrison; Richard G Sturton; Amanda J Emmons; Alison J Ford; Richard G Knowles