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药效评价Signaling of an allosteric, nanomolar potent, low molecular weight agonist for the follicle-stimulating hormone receptor.

期刊:Biochemical pharmacology发表年份:2013作者:Chris J van Koppen; Pieter M Verbost; Ruud van de Lagemaat; Willem-Jan F Karstens; Huub J J Loozen; Tanja A E van Achterberg; Monique G A van Amstel; Jolanda H G M Brands; Els J P van Doornmalen; Jesse Wat; Saskia J Mulder; Bianca C Raafs; Saskia Ver

药效评价Sphingosine 1-phosphate (S1P) receptor agonists mediate pro-fibrotic responses in normal human lung fibroblasts via S1P2 and S1P3 receptors and Smad-independent signaling.

期刊:The Journal of biological chemistry发表年份:2013作者:Katrin Sobel; Katalin Menyhart; Nina Killer; Bérengère Renault; Yasmina Bauer; Rolf Studer; Beat Steiner; Martin H Bolli; Oliver Nayler; John Gatfield

药效评价Substrate-dependent ligand inhibition of the human organic cation transporter OCT2.

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2013作者:Mathew Belzer; Mark Morales; Bhumasamudram Jagadish; Eugene A Mash; Stephen H Wright

药效评价Amelioration of autoimmune neuroinflammation by the fusion molecule Fn14·TRAIL.

期刊:Journal of neuroinflammation发表年份:2013作者:Hodaya Prinz-Hadad; Tehila Mizrachi; Michal Irony-Tur-Sinai; Tatyana B Prigozhina; Alexandra Aronin; Talma Brenner; Michal Dranitzki-Elhalel