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药效评价Asparagine deamidation dependence on buffer type, pH, and temperature.

期刊:Journal of pharmaceutical sciences发表年份:2013作者:Amanda L Pace; Rita L Wong; Yonghua Taylor Zhang; Yung-Hsiang Kao; Y John Wang

药效评价Selective CB2 agonists with anti-pruritic activity: discovery of potent and orally available bicyclic 2-pyridones.

期刊:Bioorganic & medicinal chemistry发表年份:2013作者:Ken-ichi Kusakabe; Yasuyoshi Iso; Yukio Tada; Masahiro Sakagami; Yasuhide Morioka; Nobuo Chomei; Satomi Shinonome; Keiko Kawamoto; Hideyuki Takenaka; Kiyoshi Yasui; Hiroshi Hamana; Kohji Hanasaki

药效评价Development of LC/MS/MS, high-throughput enzymatic and cellular assays for the characterization of compounds that inhibit kynurenine monooxygenase (KMO).

期刊:Journal of biomolecular screening发表年份:2013作者:Dirk Winkler; Maria Beconi; Leticia M Toledo-Sherman; Michael Prime; Andreas Ebneth; Celia Dominguez; Ignacio Muñoz-Sanjuan

药效评价Pharmacological characterization of a 5-HT1-type serotonin receptor in the red flour beetle, Tribolium castaneum.

期刊:PloS one发表年份:2013作者:Rut Vleugels; Cynthia Lenaerts; Arnd Baumann; Jozef Vanden Broeck; Heleen Verlinden