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药效评价New quinoxaline derivatives as potential MT₁ and MT₂ receptor ligands.

期刊:Molecules (Basel, Switzerland)发表年份:2012作者:Saioa Ancizu; Nerea Castrillo; Silvia Pérez-Silanes; Ignacio Aldana; Antonio Monge; Philippe Delagrange; Daniel-Henry Caignard; Silvia Galiano

药效评价Fragment screening of GPCRs using biophysical methods: identification of ligands of the adenosine A(2A) receptor with novel biological activity.

期刊:ACS chemical biology发表年份:2012作者:Dan Chen; James C Errey; Laura H Heitman; Fiona H Marshall; Adriaan P Ijzerman; Gregg Siegal

药效评价GPR35 is a target of the loop diuretic drugs bumetanide and furosemide.

期刊:Pharmacology发表年份:2012作者:Yuhua Yang; Angela Fu; Xiaosu Wu; Jeff D Reagan

药效评价In search for new chemical entities as adenosine receptor ligands: development of agents based on benzo-γ-pyrone skeleton.

期刊:European journal of medicinal chemistry发表年份:2012作者:Alexandra Gaspar; Joana Reis; Maria João Matos; Eugenio Uriarte; Fernanda Borges