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药效评价Design and application of in vivo FRET biosensors to identify protein prenylation and nanoclustering inhibitors.

期刊:Chemistry & biology发表年份:2012作者:Monika Köhnke; Steven Schmitt; Nicholas Ariotti; Andrew M Piggott; Robert G Parton; Ernest Lacey; Robert J Capon; Kirill Alexandrov; Daniel Abankwa

药效评价Evaluation of antibodies directed against human protease-activated receptor-2.

期刊:Naunyn-Schmiedeberg's archives of pharmacology发表年份:2012作者:Mark N Adams; Charles N Pagel; Eleanor J Mackie; John D Hooper

药效评价Investigations on the 4-quinolone-3-carboxylic acid motif. 6. Synthesis and pharmacological evaluation of 7-substituted quinolone-3-carboxamide derivatives as high affinity ligands for cannabinoid receptors.

期刊:European journal of medicinal chemistry发表年份:2012作者:Serena Pasquini; Maria De Rosa; Alessia Ligresti; Claudia Mugnaini; Antonella Brizzi; Nicola P Caradonna; Maria Grazia Cascio; Daniele Bolognini; Roger G Pertwee; Vincenzo Di Marzo; Federico Corelli

药效评价Intact microtubules preserve transient receptor potential vanilloid 1 (TRPV1) functionality through receptor binding.

期刊:The Journal of biological chemistry发表年份:2012作者:Barbara Storti; Ranieri Bizzarri; Francesco Cardarelli; Fabio Beltram