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药效评价Interactions of N-{[2-(4-phenyl-piperazin-1-yl)-ethyl]-phenyl}-2-aryl-2-yl-acetamides and 1-{[2-(4-phenyl-piperazin-1-yl)-ethyl]-phenyl}-3-aryl-2-yl-ureas with dopamine D2 and 5-hydroxytryptamine 5HT(1A) receptors.

期刊:Bioorganic & medicinal chemistry letters发表年份:2012作者:Vladimir Sukalovic; Djurdjica Ignjatovic; Gordana Tovilovic; Deana Andric; Kaveh Shakib; Sladjana Kostic-Rajacic; Vukic Soskic

药效评价Ranking of multidimensional drug profiling data by fractional-adjusted bi-partitional scores.

期刊:Bioinformatics (Oxford, England)发表年份:2012作者:Dorit S Hochbaum; Chun-Nan Hsu; Yan T Yang

药效评价N-substituted phenoxazine and acridone derivatives: structure-activity relationships of potent P2X4 receptor antagonists.

期刊:Journal of medicinal chemistry发表年份:2012作者:Victor Hernandez-Olmos; Aliaa Abdelrahman; Ali El-Tayeb; Diana Freudendahl; Stephanie Weinhausen; Christa E Müller

药效评价Spatial proximity between the VPAC1 receptor and the amino terminus of agonist and antagonist peptides reveals distinct sites of interaction.

期刊:FASEB journal : official publication of the Federation of American Societies for Experimental Biology发表年份:2012作者:Emilie Ceraudo; Régine Hierso; Yossan-Var Tan; Samuel Murail; Christiane Rouyer-Fessard; Pascal Nicole; Jean-Claude Robert; Nadège Jamin; Jean-Michel Neumann; Patrick Robberecht; Marc Laburthe; Alain Couvineau