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药效评价A potent and selective S1P(1) antagonist with efficacy in experimental autoimmune encephalomyelitis.

期刊:Chemistry & biology发表年份:2012作者:Jean Quancard; Birgit Bollbuck; Philipp Janser; Daniela Angst; Frédéric Berst; Peter Buehlmayer; Markus Streiff; Christian Beerli; Volker Brinkmann; Danilo Guerini; Paul A Smith; Timothy J Seabrook; Martin Traebert; Klaus Seuwen; René Hersperger; Chr

药效评价Effect of cyclosporine and rifampin on the pharmacokinetics of macitentan, a tissue-targeting dual endothelin receptor antagonist.

期刊:The AAPS journal发表年份:2012作者:Shirin Bruderer; Päivi Aänismaa; Marie-Claude Homery; Stephanie Häusler; Kyle Landskroner; Patricia N Sidharta; Alexander Treiber; Jasper Dingemanse

药效评价Urocontrin, a novel UT receptor ligand with a unique pharmacological profile.

期刊:Biochemical pharmacology发表年份:2012作者:David Chatenet; Quang-Trinh Nguyen; Myriam Létourneau; Jocelyn Dupuis; Alain Fournier

药效评价Isolation, characterization and total regioselective synthesis of the novel μO-conotoxin MfVIA from Conus magnificus that targets voltage-gated sodium channels.

期刊:Biochemical pharmacology发表年份:2012作者:Irina Vetter; Zoltan Dekan; Oliver Knapp; David J Adams; Paul F Alewood; Richard J Lewis