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药效评价Stimulus bias provides evidence for conformational constraints in the structure of a G protein-coupled receptor.

期刊:The Journal of biological chemistry发表年份:2012作者:Karen J Gregory; Patrick M Sexton; Andrew B Tobin; Arthur Christopoulos

药效评价Lead discovery, chemistry optimization, and biological evaluation studies of novel biamide derivatives as CB2 receptor inverse agonists and osteoclast inhibitors.

期刊:Journal of medicinal chemistry发表年份:2012作者:Peng Yang; Kyaw-Zeyar Myint; Qin Tong; Rentian Feng; Haiping Cao; Abdulrahman A Almehizia; Mohammed Hamed Alqarni; Lirong Wang; Patrick Bartlow; Yingdai Gao; Jürg Gertsch; Jumpei Teramachi; Noriyoshi Kurihara; Garson David Roodman; Tao Cheng; Xiang-Q

药效评价Glucagon like peptide-1 receptor expression in the human thyroid gland.

期刊:The Journal of clinical endocrinology and metabolism发表年份:2012作者:Belinda Gier; Peter C Butler; Chi K Lai; David Kirakossian; Matthew M DeNicola; Michael W Yeh

药效评价Gene transfer of c-met confers protection against D-galactosamine/lipopolysaccharide-induced acute liver failure.

期刊:Digestive diseases and sciences发表年份:2012作者:Chuanlong Zhu; Yuwen Li; Wenting Li; Quan Wu; Rentao Gao