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药效评价S32212, a novel serotonin type 2C receptor inverse agonist/α2-adrenoceptor antagonist and potential antidepressant: I. A mechanistic characterization.

期刊：The Journal of pharmacology and experimental therapeutics发表年份：2012作者：Mark J Millan; Clotilde Mannoury la Cour; Benjamin Chanrion; Delphine S Dupuis; Benjamin Di Cara; Valérie Audinot; Didier Cussac; Adrian Newman-Tancredi; Maud Kamal; Jean A Boutin; Ralf Jockers; Philippe Marin; Joël Bockaert; Olivier Muller; Anne Dek
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药效评价3-Substituted pyrazole analogs of the cannabinoid type 1 (CB₁) receptor antagonist rimonabant: cannabinoid agonist-like effects in mice via non-CB₁, non-CB₂ mechanism.

期刊：The Journal of pharmacology and experimental therapeutics发表年份：2012作者：Jenny L Wiley; Dana E Selley; Pinglang Wang; Rudresha Kottani; Srinivas Gadthula; Anu Mahadeven
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药效评价7-tert-Butyl-6-(4-chloro-phenyl)-2-thioxo-2,3-dihydro-1H-pyrido[2,3-d]pyrimidin-4-one, a classic polymodal inhibitor of transient receptor potential vanilloid type 1 with a reduced liability for hyperthermia, is analgesic and ameliorates visceral hyp

期刊：The Journal of pharmacology and experimental therapeutics发表年份：2012作者：Mark S Nash; Peter McIntyre; Alex Groarke; Elliot Lilley; Andrew Culshaw; Allan Hallett; Moh Panesar; Alyson Fox; Stuart Bevan
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药效评价New pyridobenzoxazepine derivatives derived from 5-(4-methylpiperazin-1-yl)-8-chloro-pyrido[2,3-b][1,5]benzoxazepine (JL13): chemical synthesis and pharmacological evaluation.

期刊：Journal of medicinal chemistry发表年份：2012作者：Jean-François Liégeois; Marine Deville; Sébastien Dilly; Cédric Lamy; Floriane Mangin; Mélissa Résimont; Frank I Tarazi
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