郑州微飒生物科技有限责任公司 咨询热线:0371-88821766
行业动态

行业动态

追踪行业前沿,洞察产业趋势

药效评价Ligustilide: a novel TRPA1 modulator.

期刊:Pflugers Archiv : European journal of physiology发表年份:2011作者:Jian Zhong; Federica Pollastro; Jean Prenen; Zhiming Zhu; Giovanni Appendino; Bernd Nilius

药效评价Discovery, synthesis, and structure-activity relationship development of a series of N-(4-acetamido)phenylpicolinamides as positive allosteric modulators of metabotropic glutamate receptor 4 (mGlu(4)) with CNS exposure in rats.

期刊:Journal of medicinal chemistry发表年份:2011作者:Darren W Engers; Julie R Field; Uyen Le; Ya Zhou; Julie D Bolinger; Rocio Zamorano; Anna L Blobaum; Carrie K Jones; Satyawan Jadhav; C David Weaver; P Jeffrey Conn; Craig W Lindsley; Colleen M Niswender; Corey R Hopkins

药效评价Kinetically controlled drug resistance: how Penicillium brevicompactum survives mycophenolic acid.

期刊:The Journal of biological chemistry发表年份:2011作者:Xin E Sun; Bjarne Gram Hansen; Lizbeth Hedstrom

药效评价Application of Ullmann and Ullmann-Finkelstein reactions for the synthesis of N-aryl-N-(1H-pyrazol-3-yl) acetamide or N-(1-aryl-1H-pyrazol-3-yl) acetamide derivatives and pharmacological evaluation.

期刊:European journal of medicinal chemistry发表年份:2011作者:Rebecca Deprez-Poulain; Nicolas Cousaert; Patrick Toto; Nicolas Willand; Benoit Deprez