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药效评价Discovery of a calcimimetic with differential effects on parathyroid hormone and calcitonin secretion.

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2011作者:Charles Henley; Yuhua Yang; James Davis; Jenny Ying Lin Lu; Sean Morony; Wei Fan; Monica Florio; Banghua Sun; Edward Shatzen; James K Pretorius; William G Richards; David J St Jean; Christopher Fotsch; Jeff D Reagan

药效评价Pharmacological profile of FK881(ASP6537), a novel potent and selective cyclooxygenase-1 inhibitor.

期刊:Biochemical pharmacology发表年份:2011作者:Junko Imanishi; Yoshiaki Morita; Eiji Yoshimi; Kanae Kuroda; Tomoko Masunaga; Kaoru Yamagami; Masako Kuno; Emi Hamachi; Satoshi Aoki; Fumie Takahashi; Katsuya Nakamura; Susumu Miyata; Yoshitaka Ohkubo; Seitaro Mutoh

药效评价Antihypertensive, insulin-sensitising and renoprotective effects of a novel, potent and long-acting angiotensin II type 1 receptor blocker, azilsartan medoxomil, in rat and dog models.

期刊:European journal of pharmacology发表年份:2011作者:Keiji Kusumoto; Hideki Igata; Mami Ojima; Ayako Tsuboi; Mitsuaki Imanishi; Fuminari Yamaguchi; Hiroki Sakamoto; Takanobu Kuroita; Naohiro Kawaguchi; Nobuhiro Nishigaki; Hideaki Nagaya

药效评价Synthesis and binding affinity of novel mono- and bivalent morphinan ligands for κ, μ, and δ opioid receptors.

期刊:Bioorganic & medicinal chemistry发表年份:2011作者:Bin Zhang; Tangzhi Zhang; Anna W Sromek; Thomas Scrimale; Jean M Bidlack; John L Neumeyer