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药效评价Discovery of non-glycoside sodium-dependent glucose co-transporter 2 (SGLT2) inhibitors by ligand-based virtual screening.

期刊:Journal of medicinal chemistry发表年份:2010作者:Jian-Sung Wu; Yi-Hui Peng; Jiun-Ming Wu; Chieh-Jui Hsieh; Szu-Huei Wu; Mohane Selvaraj Coumar; Jen-Shin Song; Jinq-Chyi Lee; Chi-Hui Tsai; Chiung-Tong Chen; Yu-Wei Liu; Yu-Sheng Chao; Su-Ying Wu

药效评价From the ganglioside GQ1balpha to glycomimetic antagonists of the myelin-associated glycoprotein (MAG).

期刊:Chimia发表年份:2010作者:Beat Ernst; Oliver Schwardt; Stefanie Mesch; Matthias Wittwer; Gianluca Rossato; Angelo Vedani

药效评价Measurement of sialic acid content is insufficient to assess bioactivity of recombinant human erythropoietin.

期刊:Biological & pharmaceutical bulletin发表年份:2010作者:Shigehiro Yanagihara; Yuya Taniguchi; Mareto Hosono; Eiji Yoshioka; Rika Ishikawa; Yoshihiro Shimada; Toshihiko Kadoya; Kazuhiro Kutsukake

药效评价Discovery of novel (S)-alpha-phenyl-gamma-amino butanamide containing CCR5 antagonists via functionality inversion approach.

期刊:Bioorganic & medicinal chemistry letters发表年份:2010作者:Hu-Shan Zhang; Dong-Zhi Feng; Li Chen; Ya-Qiu Long