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药效评价Synthesis and pharmacology of 1-methoxy analogs of CP-47,497.

期刊:Bioorganic & medicinal chemistry发表年份:2010作者:John W Huffman; Seon A Hepburn; Patricia H Reggio; Dow P Hurst; Jenny L Wiley; Billy R Martin

药效评价Inhibitors of the tyrosine kinase EphB4. Part 3: identification of non-benzodioxole-based kinase inhibitors.

期刊:Bioorganic & medicinal chemistry letters发表年份:2010作者:Catherine Bardelle; Bernard Barlaam; Nigel Brooks; Tanya Coleman; Darren Cross; Richard Ducray; Isabelle Green; Christine Lambert-van der Brempt; Annie Olivier; Jon Read

药效评价Synthesis of cycloalkane-annelated 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines and their evaluation as 5-HT6 receptor antagonists.

期刊:Bioorganic & medicinal chemistry letters发表年份:2010作者:Alexandre V Ivachtchenko; Dmitri E Dmitriev; Elena S Golovina; Elena S Dubrovskaya; Madina G Kadieva; Angela G Koryakova; Volodymyr M Kysil; Oleg D Mitkin; Sergey E Tkachenko; Ilya M Okun; Anton A Vorobiov

药效评价Development of a GPR23 cell-based β-lactamase reporter assay.

期刊:Methods in enzymology发表年份:2010作者:Paul H Lee; Bonnie J Hanson