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药效评价[Construction and evaluation of non-specific targeting cationic polymer lipid liposomes].

期刊:Yao xue xue bao = Acta pharmaceutica Sinica发表年份:2010作者:Tao Chen; Ru-tao Wang; Zhao Wang; Ting-li Lu; Wen Zhao

药效评价Exploration of the amine terminus in a novel series of 1,2,4-triazolo-3-yl-azabicyclo[3.1.0]hexanes as selective dopamine D3 receptor antagonists.

期刊:Journal of medicinal chemistry发表年份:2010作者:Fabrizio Micheli; Luca Arista; Barbara Bertani; Simone Braggio; Anna Maria Capelli; Susanna Cremonesi; Romano Di-Fabio; Giacomo Gelardi; Gabriella Gentile; Carla Marchioro; Alessandra Pasquarello; Stefano Provera; Giovanna Tedesco; Luca Tarsi; Silvia

药效评价3-(2-Aminocarbonylphenyl)propanoic acid analogs as potent and selective EP3 receptor antagonists. Part 1: discovery and exploration of the carboxyamide side chain.

期刊:Bioorganic & medicinal chemistry发表年份:2010作者:Masaki Asada; Tetsuo Obitsu; Toshihiko Nagase; Motoyuki Tanaka; Yoshiyuki Yamaura; Hiroya Takizawa; Ken Yoshikawa; Kazutoyo Sato; Masami Narita; Shuichi Ohuchida; Hisao Nakai; Masaaki Toda

药效评价Subtlety of the structure-affinity and structure-efficacy relationships around a nonpeptide oxytocin receptor agonist.

期刊:Journal of medicinal chemistry发表年份:2010作者:Marie-Céline Frantz; Jordi Rodrigo; Laure Boudier; Thierry Durroux; Bernard Mouillac; Marcel Hibert