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药效评价[Nalpha-benzylTyr1,cyclo(D-Asp5,Dap8)]- dynorphin A-(1-11)NH2 cyclized in the "address" domain is a novel kappa-opioid receptor antagonist.

期刊:Journal of medicinal chemistry发表年份:2005作者:Kshitij A Patkar; Xiuzhen Yan; Thomas F Murray; Jane V Aldrich

药效评价Design and synthesis of tricyclic imidazo[4,5-b]pyridin-2-ones as corticotropin-releasing factor-1 antagonists.

期刊:Journal of medicinal chemistry发表年份:2005作者:Zhiqiang Guo; John E Tellew; Raymond S Gross; Brian Dyck; Jonathan Grey; Mustapha Haddach; Mehrak Kiankarimi; Marion Lanier; Bin-Feng Li; Zhiyong Luo; James R McCarthy; Manisha Moorjani; John Saunders; Robert Sullivan; Xiaohu Zhang; Said Zamani-Kord;

药效评价Discovery of potent, nonsystemic apical sodium-codependent bile acid transporter inhibitors (Part 2).

期刊:Journal of medicinal chemistry发表年份:2005作者:Horng-Chih Huang; Samuel J Tremont; Len F Lee; Bradley T Keller; Andrew J Carpenter; Ching-Cheng Wang; Shyamal C Banerjee; Scott R Both; Theresa Fletcher; Danny J Garland; Wei Huang; Claude Jones; Kevin J Koeller; Steve A Kolodziej; James Li; Robert

药效评价Synthesis and receptor assay of aromatic-ethynyl-aromatic derivatives with potent mGluR5 antagonist activity.

期刊:Bioorganic & medicinal chemistry发表年份:2005作者:David Alagille; Ronald M Baldwin; Bryan L Roth; Jarda T Wroblewski; Ewa Grajkowska; Gilles D Tamagnan