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药效评价Synthesis and structure-activity relationships of 2-aryl-4-oxazolylmethoxy benzylglycines and 2-aryl-4-thiazolylmethoxy benzylglycines as novel, potent PPARalpha selective activators- PPARalpha and PPARgamma selectivity modulation.

期刊:Bioorganic & medicinal chemistry letters发表年份:2010作者:Xiang-Yang Ye; Stephanie Chen; Hao Zhang; Kenneth T Locke; Kevin O'Malley; Litao Zhang; Raijit Srivastava; Bowman Miao; Daniel Meyers; Hossain Monshizadegan; Debra Search; Denise Grimm; Rongan Zhang; Jonathan Lippy; Celeste Twamley; Jodi K Muckelbaue

药效评价Detection of G protein-coupled receptor-mediated cellular response involved in cytoskeletal rearrangement using surface plasmon resonance.

期刊:Biosensors & bioelectronics发表年份:2010作者:Kexin Chen; Hideru Obinata; Takashi Izumi

药效评价Pharmacokinetics-based elucidation on disparity in clinical effectiveness between varieties of Zhi Zhu Wan, a Traditional Chinese Medical formula.

期刊:Journal of ethnopharmacology发表年份:2010作者:Hongxin Cao; Xi Chen; Hui Sun; Tetsuro Sakurai; Jue Zhou; Wenjun Sun; Haitao Lv; Xijun Wang

药效评价2-imino-thiazolidin-4-one derivatives as potent, orally active S1P1 receptor agonists.

期刊:Journal of medicinal chemistry发表年份:2010作者:Martin H Bolli; Stefan Abele; Christoph Binkert; Roberto Bravo; Stephan Buchmann; Daniel Bur; John Gatfield; Patrick Hess; Christopher Kohl; Céline Mangold; Boris Mathys; Katalin Menyhart; Claus Müller; Oliver Nayler; Michael Scherz; Gunther Schmidt;