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药效评价Investigations on the 4-quinolone-3-carboxylic acid motif. 3. Synthesis, structure-affinity relationships, and pharmacological characterization of 6-substituted 4-quinolone-3-carboxamides as highly selective cannabinoid-2 receptor ligands.

期刊:Journal of medicinal chemistry发表年份:2010作者:Serena Pasquini; Alessia Ligresti; Claudia Mugnaini; Teresa Semeraro; Lavinia Cicione; Maria De Rosa; Francesca Guida; Livio Luongo; Maria De Chiaro; Maria Grazia Cascio; Daniele Bolognini; Pietro Marini; Roger Pertwee; Sabatino Maione; Vincenzo Di M

药效评价Potentiometric biosensor for studying hydroquinone cytotoxicity in vitro.

期刊:Biosensors & bioelectronics发表年份:2010作者:Yanyan Wang; Qiang Chen; Xiangqun Zeng

药效评价Design, synthesis, biological properties, and molecular modeling investigations of novel tacrine derivatives with a combination of acetylcholinesterase inhibition and cannabinoid CB1 receptor antagonism.

期刊:Journal of medicinal chemistry发表年份:2010作者:Jos H M Lange; Hein K A C Coolen; Martina A W van der Neut; Alice J M Borst; Bob Stork; Peter C Verveer; Chris G Kruse

药效评价Schistosoma haematobium: identification of new estrogenic molecules with estradiol antagonistic activity and ability to inactivate estrogen receptor in mammalian cells.

期刊:Experimental parasitology发表年份:2010作者:Mónica Catarina Botelho; Raquel Soares; Nuno Vale; Ricardo Ribeiro; Vânia Camilo; Raquel Almeida; Rui Medeiros; Paula Gomes; José Carlos Machado; José Manuel Correia da Costa