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代谢疾病Engineering of a VPAC2 receptor peptide agonist to impart dipeptidyl peptidase IV stability and enhance in vivo glucose disposal.

期刊:Journal of medicinal chemistry发表年份:2006作者:Kevin B Clairmont; Thomas M Buckholz; Carla M Pellegrino; Joanne M Buxton; Nicole Barucci; Andrea Bell; Sha Ha; Fugang Li; Thomas H Claus; Arthur I Salhanick; Kevin J Lumb

代谢疾病Unacylated as well as acylated ghrelin promotes cell survival and inhibit apoptosis in HIT-T15 pancreatic beta-cells.

期刊:Journal of endocrinological investigation发表年份:2006作者:R Granata; F Settanni; L Trovato; S Destefanis; D Gallo; M Martinetti; E Ghigo; G Muccioli

代谢疾病Synthesis and activity of small molecule GPR40 agonists.

期刊:Bioorganic & medicinal chemistry letters发表年份:2006作者:Dulce M Garrido; David F Corbett; Kate A Dwornik; Aaron S Goetz; Thomas R Littleton; Steve C McKeown; Wendy Y Mills; Terrence L Smalley; Celia P Briscoe; Andrew J Peat

代谢疾病Bicyclic[4.1.0]heptanes as phenyl replacements for melanin concentrating hormone receptor antagonists.

期刊:Bioorganic & medicinal chemistry发表年份:2006作者:Ruo Xu; Shengjian Li; Jaroslava Paruchova; Mark D McBriar; Henry Guzik; Anandan Palani; John W Clader; Kathleen Cox; William J Greenlee; Brian E Hawes; Timothy J Kowalski; Kim O'Neill; Brian D Spar; Blair Weig; Daniel J Weston