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药效评价Discovery of a biaryl cyclohexene carboxylic acid (MK-6892): a potent and selective high affinity niacin receptor full agonist with reduced flushing profiles in animals as a preclinical candidate.

期刊:Journal of medicinal chemistry发表年份:2010作者:Hong C Shen; Fa-Xiang Ding; Subharekha Raghavan; Qiaolin Deng; Silvi Luell; Michael J Forrest; Ester Carballo-Jane; Larissa C Wilsie; Mihajlo L Krsmanovic; Andrew K Taggart; Kenneth K Wu; Tsuei-Ju Wu; Kang Cheng; Ning Ren; Tian-Quan Cai; Qing Chen; J

药效评价Investigation of the histamine H3 receptor binding site. Design and synthesis of hybrid agonists with a lipophilic side chain.

期刊:Journal of medicinal chemistry发表年份:2010作者:Makoto Ishikawa; Takashi Watanabe; Toshiaki Kudo; Fumikazu Yokoyama; Miki Yamauchi; Kazuhiko Kato; Nobukazu Kakui; Yasuo Sato

药效评价Refinement of the pharmacophore of an agonist ligand of the secretin receptor using conformationally constrained cyclic hexapeptides.

期刊:Peptides发表年份:2010作者:Maoqing Dong; Pooja Narang; Delia I Pinon; Andrew J Bordner; Laurence J Miller

药效评价Nuclear targeting of an endosomal E3 ubiquitin ligase.

期刊:Traffic (Copenhagen, Denmark)发表年份:2010作者:Jeffrey P Bocock; Stephanie Carmicle; Egbert Madamba; Ann H Erickson