药效评价Discovery of a biaryl cyclohexene carboxylic acid (MK-6892): a potent and selective high affinity niacin receptor full agonist with reduced flushing profiles in animals as a preclinical candidate.
期刊:Journal of medicinal chemistry发表年份:2010作者:Hong C Shen; Fa-Xiang Ding; Subharekha Raghavan; Qiaolin Deng; Silvi Luell; Michael J Forrest; Ester Carballo-Jane; Larissa C Wilsie; Mihajlo L Krsmanovic; Andrew K Taggart; Kenneth K Wu; Tsuei-Ju Wu; Kang Cheng; Ning Ren; Tian-Quan Cai; Qing Chen; J
