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代谢疾病Discovery of a Potent and Orally Bioavailable Melatonin Receptor Agonist.

期刊:Journal of medicinal chemistry发表年份:2021作者:Yasutaka Hoashi; Takafumi Takai; Yohei Kosugi; Masato Nakashima; Masaharu Nakayama; Keisuke Hirai; Osamu Uchikawa; Tatsuki Koike

代谢疾病Discovery of a novel series of guanidinebenzoates as gut-restricted enteropeptidase and trypsin dual inhibitors for the treatment of metabolic syndrome.

期刊:Bioorganic & medicinal chemistry letters发表年份:2021作者:Xuqing Zhang; Bin Zhu; Weimei Sun; Mina Wang; Kamal Albarazanji; Brahma Ghosh; Maxwell Cummings; James Lenhard; James Leonard; Mark Macielag; James Lanter

代谢疾病Orphan GPR116 mediates the insulin sensitizing effects of the hepatokine FNDC4 in adipose tissue.

期刊:Nature communications发表年份:2021作者:Anastasia Georgiadi; Valeria Lopez-Salazar; Rabih El- Merahbi; Rhoda Anane Karikari; Xiaochuan Ma; André Mourão; Katarina Klepac; Lea Bühler; Ana Jimena Alfaro; Isabell Kaczmarek; Adam Linford; Madeleen Bosma; Olga Shilkova; Olli Ritvos; Nobuhiro Nak

代谢疾病Is LRP2 Involved in Leptin Transport over the Blood-Brain Barrier and Development of Obesity?

期刊:International journal of molecular sciences发表年份:2021作者:Elvira S Sandin; Julica Folberth; Helge Müller-Fielitz; Claus U Pietrzik; Elisabeth Herold; Thomas E Willnow; Paul T Pfluger; Ruben Nogueiras; Vincent Prevot; Thomas Krey; Markus Schwaninger