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代谢疾病The GPCR accessory protein MRAP2 regulates both biased signaling and constitutive activity of the ghrelin receptor GHSR1a.

期刊:Science signaling发表年份:2020作者:Alix A J Rouault; Luciana K Rosselli-Murai; Ciria C Hernandez; Luis E Gimenez; Gregory G Tall; Julien A Sebag

代谢疾病Characterization of the Active Components of the Multimerized sTNFRIIAdiponectin Fusion Protein Showing Both TNFα-Antagonizing and Glucose Uptake-Promoting Activities.

期刊:Endocrine, metabolic & immune disorders drug targets发表年份:2020作者:Yao Wang; Hui Lian; Xitong Wang; Tianyu Zheng; Xiaoxiao Yu; Ruzhang Chen; Zhiyong Huang; Yinxiang Lv; Ai Zhao; Jimin Gao

代谢疾病Applicability Domains Enhance Application of PPARγ Agonist Classifiers Trained by Drug-like Compounds to Environmental Chemicals.

期刊:Chemical research in toxicology发表年份:2020作者:Zhongyu Wang; Jingwen Chen; Huixiao Hong

代谢疾病Discovery of 4-Phenylpiperidine-2-Carboxamide Analogues as Serotonin 5-HT2C Receptor-Positive Allosteric Modulators with Enhanced Drug-like Properties.

期刊:Journal of medicinal chemistry发表年份:2020作者:Eric A Wold; Erik J Garcia; Christopher T Wild; Joanna M Miszkiel; Claudia A Soto; Jianping Chen; Konrad Pazdrak; Robert G Fox; Noelle C Anastasio; Kathryn A Cunningham; Jia Zhou