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代谢疾病Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist.

期刊:Molecular pharmacology发表年份:2019作者:Robert B Laprairie; Kiran Vemuri; Edward L Stahl; Anisha Korde; Jo-Hao Ho; Travis W Grim; Tian Hua; Yiran Wu; Raymond C Stevens; Zhi-Jie Liu; Alexandros Makriyannis; Laura M Bohn

代谢疾病Discovery of a small molecule RXFP3/4 agonist that increases food intake in rats upon acute central administration.

期刊:Bioorganic & medicinal chemistry letters发表年份:2019作者:Brian DeChristopher; Soo-Hee Park; Linh Vong; Derek Bamford; Hyun-Hee Cho; Rohit Duvadie; Allison Fedolak; Christopher Hogan; Toshiyuki Honda; Pramod Pandey; Olga Rozhitskaya; Liansheng Su; Elizabeth Tomlinson; Iain Wallace

代谢疾病Dietary wood pulp-derived sterols modulation of cholesterol metabolism and gut microbiota in high-fat-diet-fed hamsters.

期刊:Food & function发表年份:2019作者:Xiang Li; Huali Wang; Tianxin Wang; Fuping Zheng; Hao Wang; Chengtao Wang

代谢疾病Discovery and biological evaluation of novel G protein-coupled receptor 119 agonists for type 2 diabetes.

期刊:Archiv der Pharmazie发表年份:2019作者:Ying Zhou; Youzhi Wang; Leilei Zhang; Chunlei Tang; Bainian Feng