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药效评价Fluorinated 9H-xanthene-9-carboxylic acid oxazol-2-yl-amides as potent, orally available mGlu1 receptor enhancers.

期刊:Bioorganic & medicinal chemistry letters发表年份:2009作者:Eric Vieira; Jörg Huwyler; Synèse Jolidon; Frédéric Knoflach; Vincent Mutel; Jürgen Wichmann

药效评价Synthesis and pharmacological evaluation of dimeric follicle-stimulating hormone receptor antagonists.

期刊:ChemMedChem发表年份:2009作者:Kimberly M Bonger; Sascha Hoogendoorn; Chris J van Koppen; Cornelis M Timmers; Herman S Overkleeft; Gijsbert A van der Marel

药效评价FLIPR assays of intracellular calcium in GPCR drug discovery.

期刊:Methods in molecular biology (Clifton, N.J.)发表年份:2009作者:Kasper B Hansen; Hans Bräuner-Osborne

药效评价Discovery of a new class of non-imidazole oxazoline-based histamine H(3) receptor (H(3)R) inverse agonists.

期刊:ChemMedChem发表年份:2009作者:Sylvain Célanire; Maikel Wijtmans; Bernard Christophe; Philippe Collart; Iwan de Esch; Donald Dassesse; Christel Delaunoy; Frédéric Denonne; Véronique Durieu; Edith Gelens; Michel Gillard; Bénédicte Lallemand; Yves Lamberty; Florence Lebon; Jean-Mari