郑州微飒生物科技有限责任公司 咨询热线:0371-88821766
行业动态

行业动态

追踪行业前沿,洞察产业趋势

药效评价Characterization of novel aryl-ether, biaryl, and fluorene aspartic acid and diaminopropionic acid analogs as potent inhibitors of the high-affinity glutamate transporter EAAT2.

期刊:Molecular pharmacology发表年份:2005作者:John Dunlop; H Beal McIlvain; Tikva A Carrick; Brian Jow; Qiang Lu; Dianne Kowal; Steven Lin; Alexander Greenfield; Cristina Grosanu; Kristi Fan; Robert Petroski; John Williams; Alan Foster; John Butera

药效评价2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.

期刊:Journal of medicinal chemistry发表年份:2005作者:Patrizia Minetti; Maria Ornella Tinti; Paolo Carminati; Massimo Castorina; Maria Assunta Di Cesare; Stefano Di Serio; Grazia Gallo; Orlando Ghirardi; Fabrizio Giorgi; Luca Giorgi; Giovanni Piersanti; Francesca Bartoccini; Giorgio Tarzia

药效评价Common features in the functional surface of scorpion beta-toxins and elements that confer specificity for insect and mammalian voltage-gated sodium channels.

期刊:The Journal of biological chemistry发表年份:2005作者:Lior Cohen; Izhar Karbat; Nicolas Gilles; Nitza Ilan; Morris Benveniste; Dalia Gordon; Michael Gurevitz

药效评价Somatostatin increases phospholipase D activity and phosphatidylinositol 4,5-bisphosphate synthesis in clonal beta cells HIT-T15.

期刊:Molecular pharmacology发表年份:2005作者:Henrique Cheng; Justin A Grodnitzky; Sirintorn Yibchok-anun; Jing Ding; Walter H Hsu