药效评价Discovery process and pharmacological characterization of 2-(S)-(4-fluoro-2-methylphenyl)piperazine-1-carboxylic acid [1-(R)-(3,5-bis-trifluoromethylphenyl)ethyl]methylamide (vestipitant) as a potent, selective, and orally active NK1 receptor antagon
期刊:Journal of medicinal chemistry发表年份:2009作者:Romano Di Fabio; Cristiana Griffante; Giuseppe Alvaro; Giorgio Pentassuglia; Domenica A Pizzi; Daniele Donati; Tino Rossi; Giuseppe Guercio; Mario Mattioli; Zadeo Cimarosti; Carla Marchioro; Stefano Provera; Laura Zonzini; Dino Montanari; Sergio Melo