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代谢疾病The Bioorthogonal Isonitrile-Chlorooxime Ligation.

期刊:Journal of the American Chemical Society发表年份:2019作者:Rebecca J B Schäfer; Mattia R Monaco; Mao Li; Alina Tirla; Pablo Rivera-Fuentes; Helma Wennemers

代谢疾病Discovery of potent, low-absorbable sodium-dependent glucose cotransporter 1 (SGLT1) inhibitor SGL5213 for type 2 diabetes treatment.

期刊:Bioorganic & medicinal chemistry发表年份:2019作者:Shoichi Kuroda; Yohei Kobashi; Takahiro Oi; Kenichi Kawabe; Fumiyasu Shiozawa; Lisa Okumura-Kitajima; Mami Sugisaki-Kitano; Fusayo Io; Koji Yamamoto; Hiroyuki Kakinuma

代谢疾病Molecular Basis of Action of a Small-Molecule Positive Allosteric Modulator Agonist at the Type 1 Cholecystokinin Holoreceptor.

期刊:Molecular pharmacology发表年份:2019作者:Aditya J Desai; Ingrid Mechin; Karthigeyan Nagarajan; Celine Valant; Denise Wootten; Polo C H Lam; Andrew Orry; Ruben Abagyan; Anil Nair; Patrick M Sexton; Arthur Christopoulos; Laurence J Miller

代谢疾病Evaluation of Amides, Carbamates, Sulfonamides, and Ureas of 4-Prop-2-ynylidenecycloalkylamine as Potent, Selective, and Bioavailable Negative Allosteric Modulators of Metabotropic Glutamate Receptor 5.

期刊:Journal of medicinal chemistry发表年份:2019作者:Davide Graziani; Silvia Caligari; Elisa Callegari; Carlo De Toma; Matteo Longhi; Fabio Frigerio; Roberto Dilernia; Sergio Menegon; Luca Pinzi; Lorenza Pirona; Valerio Tazzari; Anna Elisa Valsecchi; Giulio Vistoli; Giulio Rastelli; Carlo Riva