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药效评价Electrostatically mediated liposome fusion and lipid exchange with a nanoparticle-supported bilayer for control of surface charge, drug containment, and delivery.

期刊:Journal of the American Chemical Society发表年份:2009作者:Juewen Liu; Xingmao Jiang; Carlee Ashley; C Jeffrey Brinker

药效评价Synthesis, potency, and in vivo evaluation of 2-piperazin-1-ylquinoline analogues as dual serotonin reuptake inhibitors and serotonin 5-HT1A receptor antagonists.

期刊:Journal of medicinal chemistry发表年份:2009作者:Dahui Zhou; Gary P Stack; Jennifer Lo; Amedeo A Failli; Deborah A Evrard; Boyd L Harrison; Nicole T Hatzenbuhler; Megan Tran; Susan Croce; Soo Yi; Jeannette Golembieski; Geoffrey A Hornby; Margaret Lai; Qian Lin; Lee E Schechter; Deborah L Smith; Ada

药效评价Nonpeptide urotensin-II receptor antagonists: a new ligand class based on piperazino-phthalimide and piperazino-isoindolinone subunits.

期刊:Journal of medicinal chemistry发表年份:2009作者:Edward C Lawson; Diane K Luci; Shyamali Ghosh; William A Kinney; Charles H Reynolds; Jenson Qi; Charles E Smith; Yuanping Wang; Lisa K Minor; Barbara J Haertlein; Tom J Parry; Bruce P Damiano; Bruce E Maryanoff

药效评价Differential regulation of muscarinic M1 receptors by orthosteric and allosteric ligands.

期刊:BMC pharmacology发表年份:2009作者:Christopher N Davis; Stefania Risso Bradley; Hans H Schiffer; Mikael Friberg; Kristian Koch; Bo-Ragnar Tolf; Douglas W Bonhaus; Jelveh Lameh