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药效评价The effect of assay formats on the estimation of melanocortin agonist affinity and efficacy using the operation model of agonism.

期刊:European journal of pharmacology发表年份:2009作者:Sylvie Simon; Tim J Young; Sarah A Nickolls

药效评价Effect of route of administration of human recombinant factor VIII on its immunogenicity in Hemophilia A mice.

期刊:Journal of pharmaceutical sciences发表年份:2009作者:Aaron Peng; Puneet Gaitonde; Matthew P Kosloski; Razvan D Miclea; Prashant Varma; Sathy V Balu-Iyer

药效评价Optimization of 2-piperidin-4-yl-acetamides as melanin-concentrating hormone receptor 1 (MCH-R1) antagonists: Designing out hERG inhibition.

期刊:Bioorganic & medicinal chemistry letters发表年份:2009作者:Susanne Berglund; Bryan J Egner; Henrik Gradén; Joakim Gradén; David G A Morgan; Tord Inghardt; Fabrizio Giordanetto

药效评价Synthetic small-molecule prohormone convertase 2 inhibitors.

期刊:Molecular pharmacology发表年份:2009作者:Dorota Kowalska; Jin Liu; Jon R Appel; Akihiko Ozawa; Adel Nefzi; Robert B Mackin; Richard A Houghten; Iris Lindberg