郑州微飒生物科技有限责任公司 咨询热线:0371-88821766
行业动态

行业动态

追踪行业前沿,洞察产业趋势

药效评价Comparative pharmacology of adrenergic alpha(2C) receptors coupled to Ca(2+) signaling through different Galpha proteins.

期刊:Neurochemistry international发表年份:2009作者:Dalma Kurko; Zsófia Bekes; Anikó Gere; Andrea Baki; András Boros; Sándor Kolok; Gyula Bugovics; József Nagy; Zsolt Szombathelyi; Györgyi Ignácz-Szendrei

药效评价Characterization of a cannabinoid CB2 receptor-selective agonist, A-836339 [2,2,3,3-tetramethyl-cyclopropanecarboxylic acid [3-(2-methoxy-ethyl)-4,5-dimethyl-3H-thiazol-(2Z)-ylidene]-amide], using in vitro pharmacological assays, in vivo pain models,

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2009作者:Betty B Yao; Gin Hsieh; Anthony V Daza; Yihong Fan; George K Grayson; Tiffany Runyan Garrison; Odile El Kouhen; Bradley A Hooker; Madhavi Pai; Erica J Wensink; Anita K Salyers; Prasant Chandran; Chang Z Zhu; Chengmin Zhong; Keith Ryther; Megan E Gall

药效评价Pyrido[2,3-e]-1,2,4-triazolo[4,3-a]pyrazin-1-one as a new scaffold to develop potent and selective human A3 adenosine receptor antagonists. Synthesis, pharmacological evaluation, and ligand-receptor modeling studies.

期刊:Journal of medicinal chemistry发表年份:2009作者:Vittoria Colotta; Ombretta Lenzi; Daniela Catarzi; Flavia Varano; Guido Filacchioni; Claudia Martini; Letizia Trincavelli; Osele Ciampi; Anna Maria Pugliese; Chiara Traini; Felicita Pedata; Erika Morizzo; Stefano Moro

药效评价Effects of beta3-adrenergic receptor activation on rat urinary bladder hyperactivity induced by ovariectomy.

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2009作者:F Aura Kullmann; Brian J Limberg; Debra E Artim; Mansi Shah; Thomas R Downs; Dan Contract; John Wos; Jan S Rosenbaum; William C de Groat