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药效评价In vitro and in vivo pharmacological characterization of PF-01354082, a novel partial agonist selective for the 5-HT(4) receptor.

期刊:European journal of pharmacology发表年份:2009作者:Tadayoshi Mikami; Tohru Komada; Hiromi Sugimoto; Keiko Suzuki; Takashi Ohmi; Naoji Kimura; Rie Naganeo; Eriko Nakata; Keigo Nakatani; Tetsuo Toga; Hiroyuki Eda; Minoru Sakakibara

药效评价[N-methyl-3H3]AZ10419369 binding to the 5-HT1B receptor: in vitro characterization and in vivo receptor occupancy.

期刊:The Journal of pharmacology and experimental therapeutics发表年份:2009作者:Donna L Maier; Cindy Sobotka-Briner; Min Ding; Mark E Powell; Qiaoling Jiang; Geraldine Hill; J Richard Heys; Charles S Elmore; M Edward Pierson; Ladislav Mrzljak

药效评价Effect of a novel NOP receptor agonist (SCH 225288) on guinea pig irritant-evoked, feline mechanically induced and canine infectious tracheobronchitis cough.

期刊:Pharmacology发表年份:2009作者:Robbie L McLeod; Deen B Tulshian; Ginny D Ho; Xiomara Fernandez; Donald C Bolser; Leonard E Parra; Jennifer C Zimmer; Christine H Erickson; Ahmad B Fawzi; Huchappa Jayappa; Craig Lehr; Jason Erskine; April Smith-Torhan; Hongtao Zhang; John A Hey

药效评价Evaluating cellular impedance assays for detection of GPCR pleiotropic signaling and functional selectivity.

期刊:Journal of biomolecular screening发表年份:2009作者:Matthew F Peters; Clay W Scott