其他Novel human adenosine receptor antagonists based on the 7-amino-thiazolo[5,4-d]pyrimidine scaffold. Structural investigations at the 2-, 5- and 7-positions to enhance affinity and tune selectivity.
期刊:Bioorganic & medicinal chemistry letters发表年份:2019作者:Flavia Varano; Daniela Catarzi; Matteo Falsini; Diego Dal Ben; Michela Buccioni; Gabriella Marucci; Rosaria Volpini; Vittoria Colotta
期刊:Proceedings of the National Academy of Sciences of the United States of America发表年份:2019作者:Andreas Geissner; Anika Reinhardt; Christoph Rademacher; Timo Johannssen; João Monteiro; Bernd Lepenies; Michel Thépaut; Franck Fieschi; Jana Mrázková; Michaela Wimmerova; Frank Schuhmacher; Sebastian Götze; Dan Grünstein; Xiaoqiang Guo; Heung Sik Ha