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其他Cis-activation in the Notch signaling pathway.

期刊:eLife发表年份:2019作者:Nagarajan Nandagopal; Leah A Santat; Michael B Elowitz

其他Novel human adenosine receptor antagonists based on the 7-amino-thiazolo[5,4-d]pyrimidine scaffold. Structural investigations at the 2-, 5- and 7-positions to enhance affinity and tune selectivity.

期刊:Bioorganic & medicinal chemistry letters发表年份:2019作者:Flavia Varano; Daniela Catarzi; Matteo Falsini; Diego Dal Ben; Michela Buccioni; Gabriella Marucci; Rosaria Volpini; Vittoria Colotta

其他Microbe-focused glycan array screening platform.

期刊:Proceedings of the National Academy of Sciences of the United States of America发表年份:2019作者:Andreas Geissner; Anika Reinhardt; Christoph Rademacher; Timo Johannssen; João Monteiro; Bernd Lepenies; Michel Thépaut; Franck Fieschi; Jana Mrázková; Michaela Wimmerova; Frank Schuhmacher; Sebastian Götze; Dan Grünstein; Xiaoqiang Guo; Heung Sik Ha

其他Discovery of novel 4-phenyl-2-(pyrrolidinyl)nicotinamide derivatives as potent Nav1.1 activators.

期刊:Bioorganic & medicinal chemistry letters发表年份:2019作者:Tohru Miyazaki; Masanori Kawasaki; Atsushi Suzuki; Yuki Ito; Akio Imanishi; Takamitsu Maru; Tomohiro Kawamoto; Tatsuki Koike