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心血管疾病Extracellular Loop 2 of the Adenosine A1 Receptor Has a Key Role in Orthosteric Ligand Affinity and Agonist Efficacy.

期刊:Molecular pharmacology发表年份:2016作者:Anh T N Nguyen; Jo-Anne Baltos; Trayder Thomas; Toan D Nguyen; Laura López Muñoz; Karen J Gregory; Paul J White; Patrick M Sexton; Arthur Christopoulos; Lauren T May

心血管疾病Discovery of novel N,N-3-phenyl-3-benzylaminopropionanilides as potent inhibitors of cholesteryl ester transfer protein in vivo.

期刊:Bioorganic & medicinal chemistry发表年份:2016作者:Honglei Xie; Yiqun Li; Changlin Bai; Ruifeng Wang; Chunchi Liu; Chenzhou Hao; Bin Lin; Maosheng Cheng; Dongmei Zhao

心血管疾病S-nitrosylation regulates VE-cadherin phosphorylation and internalization in microvascular permeability.

期刊:American journal of physiology. Heart and circulatory physiology发表年份:2016作者:Anita Guequén; Rodrigo Carrasco; Patricia Zamorano; Lorena Rebolledo; Pia Burboa; José Sarmiento; Mauricio P Boric; Adam Korayem; Walter N Durán; Fabiola A Sánchez

心血管疾病Potent and Selective Agonists of Sphingosine 1-Phosphate 1 (S1P1): Discovery and SAR of a Novel Isoxazole Based Series.

期刊:Journal of medicinal chemistry发表年份:2016作者:Scott H Watterson; Junqing Guo; Steve H Spergel; Charles M Langevine; Robert V Moquin; Ding Ren Shen; Melissa Yarde; Mary Ellen Cvijic; Dana Banas; Richard Liu; Suzanne J Suchard; Kathleen Gillooly; Tracy Taylor; Sandra Rex-Rabe; David J Shuster; Kim