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其他The 1,2,4-Triazolo[4,3-a]pyrazin-3-one as a Versatile Scaffold for the Design of Potent Adenosine Human Receptor Antagonists. Structural Investigations to Target the A2A Receptor Subtype.

期刊:Journal of medicinal chemistry发表年份:2017作者:Matteo Falsini; Lucia Squarcialupi; Daniela Catarzi; Flavia Varano; Marco Betti; Diego Dal Ben; Gabriella Marucci; Michela Buccioni; Rosaria Volpini; Teresa De Vita; Andrea Cavalli; Vittoria Colotta

其他Discovery and optimization of 3-(4-aryl/heteroarylsulfonyl)piperazin-1-yl)-6-(piperidin-1-yl)pyridazines as novel, CNS penetrant pan-muscarinic antagonists.

期刊:Bioorganic & medicinal chemistry letters发表年份:2017作者:Aaron M Bender; Rebecca L Weiner; Vincent B Luscombe; Sonia Ajmera; Hyekyung P Cho; Sichen Chang; Xiaoyan Zhan; Alice L Rodriguez; Colleen M Niswender; Darren W Engers; Thomas M Bridges; P Jeffrey Conn; Craig W Lindsley

其他Cell type-selective imaging and profiling of newly synthesized proteomes by using puromycin analogues.

期刊:Chemical communications (Cambridge, England)发表年份:2017作者:Shubo Du; Danyang Wang; Jun-Seok Lee; Bo Peng; Jingyan Ge; Shao Q Yao

其他Cellular uptake pathways of sepiolite nanofibers and DNA transfection improvement.

期刊:Scientific reports发表年份:2017作者:Fidel Antonio Castro-Smirnov; Jeanne Ayache; Jean-Rémi Bertrand; Elodie Dardillac; Eric Le Cam; Olivier Piétrement; Pilar Aranda; Eduardo Ruiz-Hitzky; Bernard S Lopez