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药效评价Monitoring of chloride and activity of glycine receptor channels using genetically encoded fluorescent sensors.

期刊:Philosophical transactions. Series A, Mathematical, physical, and engineering sciences发表年份:2008作者:Marat Mukhtarov; Olga Markova; Eleonore Real; Yves Jacob; Svetlana Buldakova; Piotr Bregestovski

药效评价Discovery of a novel series of benzoic acid derivatives as potent and selective human beta3 adrenergic receptor agonists with good oral bioavailability. 3. Phenylethanolaminotetraline (PEAT) skeleton containing biphenyl or biphenyl ether moiety.

期刊:Journal of medicinal chemistry发表年份:2008作者:Masashi Imanishi; Yutaka Nakajima; Yasuyo Tomishima; Hitoshi Hamashima; Kenichi Washizuka; Minoru Sakurai; Shigeo Matsui; Emiko Imamura; Koji Ueshima; Takao Yamamoto; Nobuhiro Yamamoto; Hirofumi Ishikawa; Keiko Nakano; Naoko Unami; Kaori Hamada; Yasu

药效评价Electrospray ionization mass spectrometry and exogenous heavy isotope-labeled lipid species provide detailed information on aminophospholipid acyl chain remodeling.

期刊:The Journal of biological chemistry发表年份:2008作者:Ville Kainu; Martin Hermansson; Pentti Somerharju

药效评价Discovery of a novel competitive inhibitor of PTP1B by high-throughput screening.

期刊:Acta pharmacologica Sinica发表年份:2008作者:Lei Shi; Hai-ping Yu; Yue-yang Zhou; Jun-qin Du; Qiang Shen; Jing-ya Li; Jia Li